一般注記Part A. Concepts -- 1. The drug discovery process -- 2. Drug synthesis -- 3. Retrosynthesis -- 4. Cyclic systems in drug synthesis -- 5. The synthesis of chiral drugs -- 6. Combinatorial and parallel synthesis -- Part B. Applications of drug synthesis in the drug development process -- 7. Synthesis of lead compounds -- 8. Analogue synthesis in drug design -- 9. Synthesis of natural products and their analogues -- 10. Chemical and process development -- 11. Synthesis of isotopically labelled compounds -- Part C. Design and synthesis of selected antibacterial agents -- 12. Design and synthesis of tetracyclines -- 13. Enthromycin and macrolide antibacterial agents -- 14. Quinolones and fluoroquinolones.